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RVX-208

 

CAS: 1044870-39-4

 

Chemical Name: Apabetalone; RVX-000222; 2-​[4-​(2-​Hydroxyethoxy)​-​3,​5-​dimethylphenyl]​-​5,​7-​dimethoxy-​3H-​quinazolin-​4-​one; 2-​[4-​(2-​Hydroxyethoxy)​-​3,​5-​dimethylphenyl]​-​5,​7-​dimethoxyquinazolin-​4(3H)​-​one

 

 

GLXC-04211        Cat No: GLXC-04211

 

 

Purity:               > 98% (HPLC)

Storage:             Refrigerator (4 °C)

 


Product Description:

Novel inhibitor of BET transcriptional regulators with selectivity for the second bromodomain (BD2)

 

References:

1) https://www.mdpi.com/1422-0067/21/11/4113

2) https://www.futuremedicine.com/doi/full/10.2217/fca-2020-0017?url_ver=Z39.88-2003&rfr_id=ori%3Arid%3Acrossref.org&rfr_dat=cr_pub++0pubmed&

3) https://jamanetwork.com/journals/jama/article-abstract/2763951

 

Analytical data click for PDF file

 

 

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