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CAS: 2376137-05-0
Chemical Name: 4-Amino-N-((S)-1-(4-chlorophenyl)-3-(4-(11-(((S)-1-((2S,4R)-4-hydroxy-2-((4-(4-methylthiazol-5-yl)benzyl)carbamoyl)pyrrolidin-1-yl)-3,3-dimethyl-1-oxobutan-2-yl)amino)-11-oxoundecanoyl)piperazin-1-yl)propyl)-1-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)piperidine-4-carboxamide
Purity: >98% (HPLC)
Novel degrader of AKT, selectively inhibiting the growth of PI3K/PTEN pathway-mutant cancers with wild-type KRAS and BRAF
References:
https://pubmed.ncbi.nlm.nih.gov/?term=MS21+degrader&sort=date
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