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JAK1-IN-38a

 

CAS: N/A

 

Chemical Name: 4-(((2S,4S)-1-(4-Chlorobenzyl)-2-methylpiperidin-4-yl)amino)-N-methyl-1H-pyrrolo[2,3-b]pyridine-5-carboxamide

 

 
GLXC-23535For Lab R&D Uses Only
        Cat No: GLXC-23535

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Novel highly potent JAK1-selective inhibitor, exhibiting excellent selectivity over JAK2, JAK3, and TYK2 (IC50: JAK1 0.145 nM; JAK2 2.94 nM; JAK3 2.31 nM; TYK2 8.17 nM)

 

Ref: https://pubs.acs.org/doi/10.1021/acs.jmedchem.0c01026

 

Analytical data click for PDF file

 

 

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