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Glixx Laboratorie
CAS: N/A
Chemical Name: 4-(((2S,4S)-1-(4-Chlorobenzyl)-2-methylpiperidin-4-yl)amino)-N-methyl-1H-pyrrolo[2,3-b]pyridine-5-carboxamide
Purity: >98% (HPLC)
Novel highly potent JAK1-selective inhibitor, exhibiting excellent selectivity over JAK2, JAK3, and TYK2 (IC50: JAK1 0.145 nM; JAK2 2.94 nM; JAK3 2.31 nM; TYK2 8.17 nM)
Ref: https://pubs.acs.org/doi/10.1021/acs.jmedchem.0c01026
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