Glixx Laboratories Inc
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Glixx Laboratorie
CAS: N/A
Chemical Name: AZ12908010; N-[5-[2-(3,5-Dimethoxyphenyl)ethyl]-2H-pyrazol-3-yl]-4-(1-ethylpiperidin-4-yl)benzamide
Purity: >98% (HPLC)
Novel FGFR inhibitor, completely inhibiting FGFR-1 and significantly inhibiting FGFR-4 signaling at 100 nmol/L, inhibiting extracellular signal–regulated kinase (ERK) phosphorylation and invasion in PNT1a cells expressing FGFR-1 and FGFR-4 and all prostate cancer cell lines tested
References:
https://molpharm.aspetjournals.org/content/83/4/882.long
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