Glixx Laboratories Inc

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GSK114

 

CAS: 1301760-19-9 (free base: 1301761-96-5)

 

Chemical Name: 3-[(6,7-Dimethoxy-4-quinazolinyl)amino]-4-(dimethylamino)-N-methyl-benzenesulfonamide dihydrochloride

 

 
GLXC-15820For Lab R&D Uses Only
        Cat No: GLXC-15820

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Novel selective inhibitor for elucidating the biological role of TNNI3K, displaying significant bias (40-fold) for TNNI3K over B-Raf, exceptional broad spectrum kinase selectivity, and adequate oral exposure to enable its use in cellular and in vivo studies

 

Ref: https://www.sciencedirect.com/science/article/pii/S0960894X16305194?via%3Dihub

 

Analytical data click for PDF file

 

 

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