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CAS: N/A
Chemical Name: (R)-4-((5-(Cyclohexylmethyl)-4-ethyl-1-methyl-4,5-dihydro-[1,2,4]triazolo[4,3-f]pteridin-7-yl)amino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide
Purity: >98% (HPLC)
Novel dual BRD4 and PLK1 inhibitor (IC50 values of 109 and 22 nM, respectively), showing strong antiproliferative activity against cancer cells
References:
1) https://onlinelibrary.wiley.com/doi/10.1002/cbdv.202100519
2) https://www.sciencedirect.com/science/article/abs/pii/S0223523421007716
3) https://mct.aacrjournals.org/content/19/6/1221.long
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