Glixx Laboratories Inc

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IHCH-3064

 

CAS: N/A

 

Chemical Name: 4-(2-(5-Amino-2-(furan-2-yl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-7-yl)ethyl)-N-(2-aminophenyl)benzamide

 

 
GLXC-24890For Lab R&D Uses Only
        Cat No: GLXC-24890

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Novel dual A2AR antagonist and histone deacetylase (HDAC) inhibitor, exhibiting potent binding to A2AR (Ki = 2.2 nM) and selective inhibition of HDAC1 (IC50 = 80.2 nM), with good antiproliferative activity against tumor cell lines in vitro

 

Ref: https://pubs.acs.org/doi/10.1021/acs.jmedchem.1c01155

 

Analytical data click for PDF file

 

 

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