Glixx Laboratories Inc
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Glixx Laboratorie
CAS: 2260886-64-2
Chemical Name: N-((1r,4r)-4-(3-(2-chlorophenyl)-7-((3-methyl-4-(4-methylpiperazin-1-yl)phenyl)amino)-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2H)-yl)cyclohexyl)propionamide
Purity: >98% (HPLC)
Novel highly potent EGFRC797S inhibitor (IC50: 5.8 nM), also potently suppressing EGFRL858R/T790M (IC50:30.5 nM) and EGFRWT (IC50: 6.8 nM)
Ref: https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6231186/
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