Glixx Laboratories Inc

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Glixx Laboratorie

 

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RL-338

 

CAS: N/A

 

Chemical Name: 3-[4-(2-Fluoro-4-methoxyphenoxy)piperidin-1-yl]-N-propan-2-ylpyrazino[2,3-d]pyridazin-2-amine

 

 
GLXC-23917For Lab R&D Uses Only
        Cat No: GLXC-23917

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Novel potent and highly selective GPR6 inverse agonist, inhibiting GPR6 cAMP signalling in TR-FRET assays with a EC50 = 16 nM and >100 fold selectivity against GPR3 and GPR12

 

Ref: https://jpet.aspetjournals.org/content/early/2021/04/01/jpet.120.000438

 

Analytical data click for PDF file

 

 

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