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CAS: 2648855-18-7


Chemical Name: N-[(2S)-1-[(4-Cyanophenyl)amino]-4-cyclopropyl-1-oxidanylidene-butan-2-yl]-3,6,6-trimethyl-4-oxidanylidene-5,7-dihydro-1H-indole-2-carboxamide


GLXC-27055For Lab R&D Uses Only
        Cat No: GLXC-27055


Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)



Product Description:

Novel potent inhibitor of G9a/GLP (IC50 = 27 nM/53 nM), exhibiting remarkable selectivity against other related methyltransferases, dose-dependent attenuation of cellular H3K9me2 levels, and tumor growth inhibition in MOLT-4 cells in vitro, showing inhibition of tumor initiation and growth in a carcinogen-induced hepatocellular carcinoma (HCC) in vivo mouse model without overt acute toxicity




Analytical data click for PDF file



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