Glixx Laboratories Inc
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Glixx Laboratorie
CAS: 2378626-29-8
Chemical Name: 2-Chloro-1-(2-((3-(trifluoromethyl)phenyl)amino)phenyl)ethan-1-one
Purity: >98% (HPLC)
Novel covalent inhibitor of TEAD4-Yap1 protein-protein interaction in mammalian cells, blocking iTEAD transcriptional activity and inhibiting glioblastoma cell viability
References:
1) https://www.cell.com/cell-chemical-biology/fulltext/S2451-9456(18)30432-X
2) https://pubs.acs.org/doi/10.1021/acs.jmedchem.0c01275
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