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MT-802

 

CAS: 2231744-29-7

 

Chemical Name: MT802; 2-(2-(2-(4-(4-Amino-3-(4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)ethoxy)ethoxy)-N-(2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-5-yl)acetamide

 

 
GLXC-15887For Lab R&D Uses Only
        Cat No: GLXC-15887

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Novel PROTAC-mediated degrader, binding fewer off-target kinases than ibrutinib does, inducing BTK knockdown, recruiting BTK to the cereblon E3 ubiquitin ligase complex to trigger BTK ubiquitination and degradation via the proteasome

 

References:

1) https://www.sciencedirect.com/science/article/pii/S0960894X19308558

2) https://pubs.acs.org/doi/10.1021/acs.biochem.8b00391

 

Analytical data click for PDF file

 

 

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