Glixx Laboratories Inc

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Glixx Laboratorie

 

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 LY3039478

 

CAS: 1421438-81-4

 

Chemical Name: Crenigacestat; 4,4,4-Trifluoro-N-[(2S)-1-[[(7S)-5-(2-hydroxyethyl)-6-oxo-7H-pyrido[2,3-d][3]benzazepin-7-yl]amino]-1-oxopropan-2-yl]butanamide

 

 

GLXC-12323        Cat No: GLXC-12323

           For Lab R&D Uses Only

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 


Product Description:

Novel orally bioavailable, potent Notch inhibitor, reducing intrahepatic cholangiocarcinoma progression by blocking VEGFA/DLL4/MMP13 axis

 

References:

https://www.nature.com/articles/s41418-020-0505-4https://mcr.aacrjournals.org/content/18/1/57.long

https://www.sciencedirect.com/science/article/abs/pii/S0006291X19308393

 

Analytical data click for PDF file

 

 

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