Glixx Laboratories Inc
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Glixx Laboratorie
CAS: 2093408-03-6
Chemical Name: Isox-Cha-Chg-A-R-NH2; N-((6S,9S,12S,15S)-1-Amino-6-carbamoyl-12,16-dicyclohexyl-1-imino-9-methyl-8,11,14-trioxo-2,7,10,13-tetraazahexadecan-15-yl)isoxazole-5-carboxamide
Purity: >98% (HPLC)
Novel potent Protease activated receptor 2 (PAR2) ERK-biased agonist (EC50 2 nM, ERK1/2; EC50 80 nM, Ca2+)
Ref: https://pubs.acs.org/doi/10.1021/acschembio.6b01088
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