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CAS: 2821803-61-4
Chemical Name: 2-(4-(6-((6-Acetyl-8-cyclopentyl-5-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl)amino)pyridin-3-yl)piperazin-1-yl)-N-((1-(4-(2-amino-4-chloro-7-((4-methoxy-3,5-dimethylpyridin-2-yl)methyl)-7H-pyrrolo[2,3-d]pyrimidin-5-yl)but-3-yn-1-yl)-1H-1,2,3-triazol-4-yl)methyl)acetamide
Purity: >98% (HPLC)
Novel heat shock protein 90 (HSP90)-mediated targeting chimeras (HEMTAC), inducing intracellular CDK4/6 protein degradation
Reference:
https://pubs.acs.org/doi/10.1021/acs.jmedchem.2c01648
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