Glixx Laboratories Inc
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Glixx Laboratorie
CAS: N/A
Chemical Name: (2S,4R)-4-Hydroxy-1-((S)-2-(2-(2-(4-(3-((4-((4-(1-isopropyl-2-methyl-1H-imidazol-5-yl)pyrimidin-2-yl)amino)phenyl)sulfonyl)propyl)-1H-1,2,3-triazol-1-yl)ethoxy)acetamido)-3,3-dimethylbutanoyl)-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide
Purity: >98% (HPLC)
First-in-class selective, partial CDK2 degrader against hearing loss and cancer, protecting against cisplatin ototoxicity and kainic acid excitotoxicity
Ref: https://www.sciencedirect.com/science/article/abs/pii/S022352342100698X
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