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CAS: 1950634-92-0
Chemical Name: 2-((S)-4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)-N-(8-(2-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)oxy)acetamido)octyl)-acetamide
Cat No: GLXC-10995
Purity: >98% (HPLC)
Storage: Refrigerator (4 °C)
Novel degrader of BET bromodomain proteins, prompting a collapse of global elongation that phenocopies CDK9 inhibition
References:
https://pubmed.ncbi.nlm.nih.gov/?term=dBET6&sort=date
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