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Glixx Laboratorie
CAS: 2765264-50-2
Chemical Name: 2-(5-Fluoropyridin-2-yl)-6,6-bis(methyl-d3)-3-(1H-pyrazolo[3,4-b]pyridin-4-yl)-6,7-dihydro-4H-pyrazolo[5,1-c][1,4]oxazine
Purity: >98% (HPLC)
Novel selective and brain-penetrant inhibitor of CSNK1D (IC50 = 2.3 nM) and CSNK1E (IC50 = 137 nM)
Reference:
https://pubs.acs.org/doi/10.1021/acsmedchemlett.3c00523
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