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CAS: N/A
Chemical Name: (2R,4R)-1-(1-(4-Chlorophenyl)-3,3-difluorocyclobutane-1-carbonyl)-4-fluoro-N-(1H-pyrazolo[4,3-b]pyridin-5-yl)pyrrolidine-2-carboxamide
Purity: >98% (HPLC)
Novel highly potent p300/CBP histone acetyltransferase (HAT) inhibitor (p300 pIC50 = 10.1 and cMyc HTRF pEC50 = 8.5)
Reference:
https://pubs.acs.org/doi/10.1021/acs.jmedchem.2c00670
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