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Glixx Laboratorie
CAS: 2766352-64-9
Chemical Name: PI3K degrader HL-8; (2R,4S)-1-((S)-2-(7-(2-(5-(6-(5-((2,4-Difluorophenyl)sulfonamido)-6-methoxypyridin-3-yl)imidazo[1,2-a]pyridin-3-yl)-1,3,4-oxadiazol-2-yl)benzamido)heptanamido)-3,3-dimethylbutanoyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide
For Lab R&D Uses Only
Purity: >98% (HPLC)
Novel PI3K degrader, showing a significant and complete degradation effect on PI3K kinase at a concentration of 10 μM within 8 h
Ref: https://www.sciencedirect.com/science/article/abs/pii/S0968089622000992
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