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BIM-46187

 

CAS: 892546-37-1

 

Chemical Name: BIM-46187; PH-064; (8S,8'S)-7,7'-[Dithiobis[(2R)-2-amino-1-oxo-3,1-propanediyl]]bis[8-(cyclohexylmethyl)-5,6,7,8-tetrahydro-2-phenyl-imidazo[1,2-a]pyrazine

 

 

GLXC-05258        Cat No: GLXC-05258

 

 

Purity:               > 98% (HPLC)

Storage:             Refrigerator (4 °C)

 


Product Description:

pan G protein inhibitor, specifically silencing Gαq proteins by "freezing" Gαq in its empty pocket conformation, a conformational intermediate along the Gα activation pathway

 

 

 

Analytical data click for PDF file

 

 

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