Glixx Laboratories Inc
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Glixx Laboratorie
CAS: 2230821-38-0
Chemical Name: SJF1528; PROTAG 1; (2S,4R)-1-((S)-2-(2-(2-(2-(4-(4-((3-Chloro-4-((3-fluorobenzyl)oxy)phenyl)amino)quinazolin-6-yl)phenoxy)ethoxy)ethoxy)acetamido)-3,3-dimethylbutanoyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide
For Lab R&D Uses Only
Purity: >98% (HPLC)
Novel potent EGFR degrader, being capable of penetrating the cell membrane, also degrading an exon-20 insertion mutant form of EGFR (ASV duplication)
Ref: https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5831399/
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