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Glixx Laboratorie
CAS: N/A
Chemical Name: N-(1-(1,1-Di(pyridin-2-yl)ethyl)-6-(1-methyl-7-oxo-6,7-dihydro-1H-pyrrolo[2,3-c]pyridin-3-yl)-1H-indol-4-yl)ethanesulfonamide
Purity: >98% (HPLC)
Novel dual BET/EP300 inhibitor that represses oncogenic KRAS and potentiates immune checkpoint inhibition in pancreatic cancer
Ref: https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8795568/
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