Glixx Laboratories Inc
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Glixx Laboratorie
CAS: 3034805-75-6
Chemical Name: 5-(4-(4-(6-((2,4-Difluorobenzyl)amino)-4-((5-methyl-1H-pyrazol-3-yl)amino)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidine-1-carbonyl)piperidin-1-yl)-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione
For Lab R&D Uses Only
Purity: >98% (HPLC)
The first selective PLK4 proteolysis targeting chimera (PROTAC) degrader, exhibiting effective PLK4 degradation, more potent inhibition of cell growth, and more efficient precision-therapeutic effect in the TRIM37-amplified MCF-7 cell line than conventional inhibitor CZS-035
Reference:
https://pubs.acs.org/doi/10.1021/acs.jmedchem.3c00505
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