Glixx Laboratories Inc

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AR PROTAC A16

 

CAS: N/A

 

Chemical Name: 4-(3-(3-(4-((2-(2-((2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)oxy)ethoxy)ethoxy)methyl)-1H-1,2,3-triazol-1-yl)propyl)-4,4-dimethyl-5-oxo-2-thioxoimidazolidin-1-yl)-2-(trifluoromethyl)benzonitrile

 

 
GLXC-24341For Lab R&D Uses Only
        Cat No: GLXC-24341

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Novel potent androgen receptor (AR) degrader, exhibiting excellent AR binding affinity (85%) and AR degradation efficacy at 30 μM

 

Ref: https://www.sciencedirect.com/science/article/abs/pii/S0968089621003394

 

Analytical data click for PDF file

 

 

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