Glixx Laboratories Inc

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iBET-BD1 dihydrochloride

 

CAS: 2451862-42-1 (free base)

 

Chemical Name: GSK778 2HCl; 4-(2-(Methoxymethyl)-1-((R)-1-phenylethyl)-8-(((S)-pyrrolidin-3-yl)methoxy)-1H-imidazo[4,5-c]quinolin-7-yl)-3,5-dimethylisoxazole dihydrochloride

 

 
GLXC-22368For Lab R&D Uses Only
        Cat No: GLXC-22368

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Novel potent and selective BD1 inhibior (IC50: BRD2 BD1: 75nM; BRD3 BD1 41nM; BRD4 BD1 41nM)

 

References:

1) https://science.sciencemag.org/content/368/6489/387

2) https://bookcafe.yuntsg.com/ueditor/jsp/upload/file/20200522/1590112787777052726.pdf

 

Analytical data click for PDF file

 

 

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