Glixx Laboratories Inc
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Glixx Laboratorie
CAS: 2451862-42-1 (free base)
Chemical Name: GSK778 2HCl; 4-(2-(Methoxymethyl)-1-((R)-1-phenylethyl)-8-(((S)-pyrrolidin-3-yl)methoxy)-1H-imidazo[4,5-c]quinolin-7-yl)-3,5-dimethylisoxazole dihydrochloride
Purity: >98% (HPLC)
Novel potent and selective BD1 inhibior (IC50: BRD2 BD1: 75nM; BRD3 BD1 41nM; BRD4 BD1 41nM)
References:
1) https://science.sciencemag.org/content/368/6489/387
2) https://bookcafe.yuntsg.com/ueditor/jsp/upload/file/20200522/1590112787777052726.pdf
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