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CAS: N/A
Chemical Name: (2S,4R)-1-((S)-3,3-Dimethyl-2-(9-(4-((4-(3-(pyridin-3-ylmethyl)ureido)phenyl)sulfonyl)piperazin-1-yl)nonanamido)butanoyl)-4-hydroxy-N-((S)-1-(4-(4-methylthiazol-5-yl)phenyl)ethyl)pyrrolidine-2-carboxamide
Purity: >98% (HPLC)
Novel highly potent nicotinamide phosphoribosyltransferase (NAMPT) degrader for efficient treatment of ovarian cancer, displayed excellent degradation activity (DC50 < 0.17 nM, Dmax > 90%) and antiproliferative potency against A2780 cells (IC50 = 1.5 nM)
Reference:
https://pubs.acs.org/doi/abs/10.1021/acs.jmedchem.2c01990
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