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CAS: N/A
Chemical Name: N-((3-(3-Fluoro-4-methoxyphenyl)-4,5-dihydroisoxazol-5-yl)methyl)acrylamide
Purity: >98% (HPLC)
Novel covalent recruiter against the E2 ubiquitin conjugating enzyme UBE2D, selectively targeting C111 without targeting the catalytic C85, not inhibiting TP53 ubiquitination activity
Reference:
https://pubs.acs.org/doi/10.1021/acschembio.3c00040
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