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CAS: N/A
Chemical Name: 3-((4-(4-(4-((1-(3-(2-((2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)amino)ethoxy)propanoyl)piperidin-4-yl)methyl)piperazin-1-yl)piperidin-1-yl)-3-methoxyphenyl)amino)-6-ethyl-5-((tetrahydro-2H-pyran-4-yl)amino)pyrazine-2-carboxamide
Purity: >98% (HPLC)
Novel potent degrader of FLT3-ITD via the ubiquitin-proteasome system and inhibiting the proliferation of FLT3-ITD mutant AML cells more effectively than gilteritinib
Reference:
https://pubs.acs.org/doi/10.1021/acsmedchemlett.2c00402
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