Glixx Laboratories Inc

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Glixx Laboratorie

 

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DC-K2in212

 

CAS: N/A

 

Chemical Name: 5-(2,4-Difluoro-3-((3-((4-fluorophenyl)carbamoyl)-1H-pyrazol-4-yl)carbamoyl)phenyl)picolinamide

 

 
GLXC-23739For Lab R&D Uses Only
        Cat No: GLXC-23739

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Novel potent CDK2 inhibitor with selectivities above 10-fold over CDK1/4/6/7/9/12 above 10-fold, displaying anti-proliferative activity against A2058 melanoma and MV4-11 leukemia cell lines and low toxicity on human normal cell lines, inhibiting CDK2-medieated phosphorylation of Rb, blocking cell cycle progression, and inducing apoptosis

 

Ref: https://www.sciencedirect.com/science/article/abs/pii/S0223523421001306

 

Analytical data click for PDF file

 

 

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