Glixx Laboratories Inc
Your exclusive source for bioactive molecules
Glixx Laboratorie
CAS: 1070790-89-4
Chemical Name: CYC065; (2R,3S)-3-((6-((2,4-Dimethylbenzyl)amino)-9-isopropyl-9H-purin-2-yl)amino)pentan-2-ol
Purity: >98% (HPLC)
Novel CDK inhibitor, targeting key pro-survival and oncogenic pathways in cancer, exhibiting improved potency and selectivity for CDK2 and CDK9 compared to seliciclib, and also displaying high selectivity across the kinome
References:
1) https://journals.plos.org/plosone/article?id=10.1371/journal.pone.0234103
2) https://www.ncbi.nlm.nih.gov/pmc/articles/PMC6059250/
3) https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5553400/
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