Glixx Laboratories Inc
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Glixx Laboratorie
CAS: 1660117-38-3
Chemical Name: BI894999; 2,4-Dimethyl-6-[6-(oxan-4-yl)-1-[(1S)-1-phenylethyl]imidazo[4,5-c]pyridin-2-yl]pyridazin-3-one
Purity: >98% (HPLC)
Novel potent and selective BET inhibitor with IC50 values for BRD4-BD1 (5 nM) and BRD4-BD2 (41 nM)
References:
1) https://www.nature.com/articles/s41388-018-0150-2
2) https://www.sciencedirect.com/science/article/pii/S0304383518301514?via%3Dihub
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