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TX1-85-1

 

CAS: 1603845-32-4

 

Chemical Name: TX-85-1; N-(5-(1-(4-(4-Acetylpiperazin-1-yl)cyclohexyl)-4-amino-1H-pyrazolo[3,4-d]pyrimidin-3-yl)-2-phenoxyphenyl)acrylamide

 

 

GLXC-05772        Cat No: GLXC-05772

 

 

Purity:               > 98% (HPLC)

Storage:             Refrigerator (4 °C)

 


Product Description:

The first selective Her3 ligand, forming a covalent bond with Cys721 located in the ATP-binding site of Her3

 

References:

1) https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4633287/

2) https://www.nature.com/articles/nchembio.1658

 

Analytical data click for PDF file

 

 

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