Glixx Laboratories Inc

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 BI-9564

 

CAS: 1883429-22-8

 

Chemical Name: 4-(4-Dimethylaminomethyl-2,5-dimethoxy-phenyl)-2-methyl-2H-[2,7]naphthyridin-1-one

 

 

GLXC-07027        Cat No: GLXC-07027

 

 

Purity:               > 98% (HPLC)

Storage:             Refrigerator (4 °C)


Product Description:

Novel BRD9/7 specific inhibitor, binding to BRD9 with a higher affinity (Kd=14 nM, ITC) than to BRD7 (Kd=239nM, ITC), being completely negative on BET family members (>100 µM by AlphaScreen) and demonstrating cellular activity by FRAP on BRD9 and BRD7 at 0.1 µM and 1 µM, respectively

 

References:

1) https://www.mdpi.com/1422-0067/18/7/1537

2) https://pubs.acs.org/doi/10.1021/acs.jmedchem.6b00550

3) https://pubs.acs.org/doi/10.1021/acs.jmedchem.5b01865

 

Analytical data click for PDF file

 

 

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