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CAS: N/A
Chemical Name: (2S,4R)-1-((R)-3-((6-(2-((S)-4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)acetamido)hexyl)thio)-2-(1-fluorocyclopropane-1-carboxamido)-3-methylbutanoyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide
Purity: >98% (HPLC)
Novel AT1 (GLXC-12072) analog, degrading proteins to E3 ubiquitin ligases
Reference:
https://www.nature.com/articles/s41589-022-01177-2
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