Glixx Laboratories Inc

               Your exclusive source for bioactive molecules

Glixx Laboratorie

 

   sales@glixxlabs.com      Toll-Free: (855)Go-Glixx   Tel: 781-333-5348    Fax: 781-333-5368 
SKLB-03220

 

CAS: 2852050‑29‑2

 

Chemical Name: 5'-Acrylamido-N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-5-(ethyl(tetrahydro-2H-pyran-4-yl)amino)-2',4-dimethyl-[1,1'-biphenyl]-3-carboxamide

 

 
GLXC-26853For Lab R&D Uses Only
        Cat No: GLXC-26853

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Novel potent and selective EZH2 covalent inhibitor, bindpng to the S-adenosylmethionine (SAM) pocket of EZH2, being highly potent for EZH2MUT, while exhibiting weak activities against other tested histone methyltransferases (HMTs) and kinases

 

Reference:

https://pubs.acs.org/doi/10.1021/acs.jmedchem.2c01370

 

Analytical data click for PDF file

 

 

Place an order!

Price & Availability





POA
 








Bulk inquiry contact:
sales@glixxlabs.com
service@glixxlabs.com