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CAS: N/A
Chemical Name: 2-((S)-4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)-N-(5-(2-(4-(2,6-dioxopiperidin-3-yl)phenoxy)acetamido)pentyl)acetamide
Purity: >98% (HPLC)
Novel BET PROTAC as a uniquely potent degrader of BET proteins
Ref: https://onlinelibrary.wiley.com/doi/10.1002/anie.202108848
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