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CAS: N/A
Chemical Name: (R)-N-((2-Amino-5-chloro-3-fluoropyridin-4-yl)(7-(4-(2-hydroxypropan-2-yl)pyridin-2-yl)benzo[b]thiophen-2-yl)methyl)cyclopropanesulfonamide
For Lab R&D Uses Only
Purity: >98% (HPLC)
Novel disrupter of glucokinase-glucokinase regulatory protein (GK-GKRP) binding, inducing GK translocation from the nucleus to the cytoplasm in rats and blood glucose reduction in mice
Ref: https://pubs.acs.org/doi/10.1021/acs.jmedchem.5b01367
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