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CAS: N/A
Chemical Name: 2-(((2R,3S,4R,5R)-5-(6-Amino-2-chloro-9H-purin-9-yl)-3-ethynyl-3,4-dihydroxytetrahydrofuran-2-yl)methoxy)-2-(4-(2-oxotetrahydropyrimidin-1(2H)-yl)benzyl)malonic acid
Purity: >98% (HPLC)
Novel orally bioavailable and highly potent CD73 inhibitor, reversing AMP-mediated suppression of CD8+ T cells and completely inhibited CD73 activity in serum samples from various cancer patients
Reference:
https://pubs.acs.org/doi/abs/10.1021/acs.jmedchem.2c01287
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