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CAS: 2573775-59-2
Chemical Name: Cbl-b-IN-3; 2-(3-((1S,3R)-3-Methyl-1-(4-methyl-4H-1,2,4-triazol-3-yl)cyclobutyl)phenyl)-6-(((S)-3-methylpiperidin-1-yl)methyl)-4-(trifluoromethyl)isoindolin-1-one
For Lab R&D Uses Only
Purity: >98% (HPLC)
Novel potent casitas B lineage lymphoma proto-oncogene-b (Cbl-b) inhibitor (IC50<1 nM)
Reference:
https://jitc.bmj.com/content/11/2/e006007.long
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