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NAH-C3-GPKK

 

CAS: N/A

 

Chemical Name: ((S)-2-((S)-1-((3-(((S)-3-Amino-3-carboxypropyl)(((2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-dihydroxytetrahydrofuran-2-yl)methyl)amino)propyl)glycyl)pyrrolidine-2-carboxamido)-6-(l2-azaneyl)hexanoyl)-L-lysine

 

 
GLXC-24173For Lab R&D Uses Only
        Cat No: GLXC-24173

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Novel potent protein N-terminal methyltransferase 1 (NTMT1) bisubstrate inhibitor (Ki, app = 7 ± 1 nM), also potently inhibiting a methyltransferase complex HemK2-Trm112 (also known as KMT9-Trm112)

 

Ref: https://www.biorxiv.org/content/10.1101/2021.04.13.439666v1

 

Analytical data click for PDF file

 

 

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