Glixx Laboratories Inc

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 AVN-101

 

CAS: 1061354-48-0

 

Chemical Name: 2,8-Dimethyl-5-phenethyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole hydrochloride

 

 

GLXC-08795        Cat No: GLXC-08795

 

 

Purity:               > 98% (HPLC)

Storage:             Refrigerator (4 °C)

 


Product Description:

Highly potent 5-HT7 receptor antagonist (Ki=153 pM) with slightly lesser potency toward 5-HT6, 5-HT2A, and 5HT-2C receptors (Ki=1.2-2.0 nM), also exhibiting a rather high affinity toward histamine H1 (Ki=0.58 nM) and adrenergic alpha2A, alpha2B, and alpha2C (Ki=0.41-3.6 nM) receptors.

 

Analytical data click for PDF file

 

 

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