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CAS: 2828438-38-4
Chemical Name: 3-(2,6-Dichloro-3,5-dimethoxyphenyl)-1-(6-((4-(4-(1-(2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-5-yl)piperidine-4-carbonyl)piperazin-1-yl)phenyl)amino)pyrimidin-4-yl)-1-methylurea
For Lab R&D Uses Only
Purity: >98% (HPLC)
Novel efficient and selective FGFR2 proteolysis-targeting degrader, preferentially internalizing and degrading membrane-bound FGFR2 among the four FGFR isoforms
Reference:
https://pubs.acs.org/doi/10.1021/acs.jmedchem.3c00150
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