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Glixx Laboratorie
CAS: 2737222-94-3
Chemical Name: N-(4'-((5-(((S)-1-((2S,4R)-4-Hydroxy-2-((4-(4-methylthiazol-5-yl)benzyl)carbamoyl)pyrrolidin-1-yl)-3,3-dimethyl-1-oxobutan-2-yl)amino)-5-oxopentyl)carbamoyl)-4-(4-methylpiperazin-1-yl)-[1,1'-biphenyl]-3-yl)-6-oxo-4-(trifluoromethyl)-1,6-dihydropyridine-3-carboxamide
For Lab R&D Uses Only
Purity: >98% (HPLC)
The first potent and selective degrader probe for the WDR5 protein with a KD (ITC) of 18 nM
Reference:
https://pubs.acs.org/doi/10.1021/acs.jmedchem.1c00146
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