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CAS: N/A
Chemical Name: 2-((2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)oxy)-N-(2-(2-(2-(4-(5-(2-(5-isopropyl-2-methylphenoxy)pyrimidin-4-yl)-4-(4-(trifluoromethyl)phenyl)-1H-imidazol-1-yl)piperidin-1-yl)ethoxy)ethoxy)ethyl)acetamide
Purity: >98% (HPLC)
Novel selective N-terminal BRD4 bromodomain-targeted degrader (DC50 = 280 nM), upregulating BRD2/3
Ref: https://pubs.acs.org/doi/10.1021/acsmedchemlett.2c00300
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