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Glixx Laboratorie
CAS: 1403679-33-3
Chemical Name: 5-(2-Amino-4-pyrimidinyl)-2-[2-chloro-5-(trifluoromethyl)phenyl]-1H-pyrrole-3-carboxamide
Cat No: GLXC-12369
Purity: >98% (HPLC)
Storage: Refrigerator (4 °C)
Novel JAK2 inhibitor, displaying significant tumor growth inhibition in SET-2 xenograft tumor model, with a mechanism of action confirmed in vivo by typical modulation of known biomarkers, and with a favorable pharmacokinetic and safety profile
Reference:
https://www.sciencedirect.com/science/article/abs/pii/S0968089614004714
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