Glixx Laboratories Inc
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Glixx Laboratorie
CAS: 1895049-20-3
Chemical Name: GSK525762C; I-BET-762 besylate; 2-[(4S)-6-(4-Chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-ethylacetamide besylate
Purity: >98% (HPLC)
Novel inhibitor of the BET (Bromodomain and Extra-Terminal) family of bromodomain-containing proteins with potential antineoplastic activity
References:
1) https://accp1.onlinelibrary.wiley.com/doi/full/10.1002/jcph.1711
2) https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7165800/
3) https://onlinelibrary.wiley.com/doi/abs/10.1002/pbc.28267
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