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Glixx Laboratorie
CAS: N/A
Chemical Name: 3-(2,6-Dichloro-3,5-dimethoxy-phenyl)-1-[1-(4-dimethylamino-but-2-enoyl)-piperidin-4-yl]-7-phenylamino-3,4-dihydro-1H-pyrimido[4,5-d]pyrimidin-2-one
Purity: >98% (HPLC)
Novel potentl and selective covalent FGFR inhibitor, inhibiting proliferation of FGFR-amplified cancer cell lines with low nM IC50 values
Ref: https://www.sciencedirect.com/science/article/abs/pii/S022352341730315X
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