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CAS: N/A
Chemical Name: (S)-4'-((5-(2-(4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)acetamido)pentyl)oxy)-N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-5-(ethyl(tetrahydro-2H-pyran-4-yl)amino)-4-methyl-[1,1'-biphenyl]-3-carboxamide
Purity: >98% (HPLC)
First-in-class dual EZH2/BRD4 inhibitor, displaying potent inhibitory activity against EZH2 and BRD4 and remarkable antiproliferative capacity against 11 solid cancer cell lines
Ref: https://pubs.acs.org/doi/10.1021/acs.jmedchem.1c01876
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