Glixx Laboratories Inc
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Glixx Laboratorie
CAS: 2222941-37-7
Chemical Name: CCS1477; (6S)-1-(3,4-Difluorophenyl)-6-[5-(3,5-dimethyl-1,2-oxazol-4-yl)-1-(4-methoxycyclohexyl)benzimidazol-2-yl]piperidin-2-one
Purity: >98% (HPLC)
Novel inhibitor of the p300/CBP conserved bromodomain, inhibiting cell proliferation in prostate cancer cell lines and decreasing AR- and C-MYC-regulated gene expression, modulating KLK3 blood levels and regulating CRPC biopsy biomarker expression
References:
https://pubmed.ncbi.nlm.nih.gov/?term=CCS-1477&sort=date
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